Friday, August 12, 2016

Rotenone Mechanism of Action


Rotenone is an odorless, colorless, apparent isoflavone acclimated as a broad-spectrum insecticide, piscicide, and pesticide. It occurs by itself in the seeds and stems of several plants, such as the jicama backcountry plant, and the roots of several associates of Fabaceae. It was the aboriginal declared affiliate of the ancestors of actinic compounds accepted as rotenoids.

Rotenone works by interfering with the electron carriage alternation in mitochondria. It inhibits the alteration of electrons from iron-sulfur centers in circuitous I to ubiquinone. This interferes with NADH during the conception of accessible cellular activity (ATP). Circuitous I is clumsy to canyon off its electron to CoQ, creating a back of electrons aural the mitochondrial matrix. Cellular oxygen is bargain to the radical, creating a acknowledging oxygen species, which can accident DNA and added apparatus of the mitochondria.

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